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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T28531 | Facinicline hydrochloride | RG3487 | 5-HT Receptor , AChR |
Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM). Facinicline hydrochloride improves cognition and sensorimot... | |||
T8593 | RU 24969 | 5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole | 5-HT Receptor |
RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors. | |||
T7350 | Nelotanserin | APD125 | 5-HT Receptor |
Nelotanserin (APD125) is a potent 5-HT2A inverse agonist(IC50 : 1.7 nM), a moderately potent 5-HT2C partial inverse agonist t(IC50 :79 nM )and a weak 5-HT2B inverse agonistt(IC50 : 791 nM). | |||
T4266 | LY334370 | LY 334370 | 5-HT Receptor |
LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM | |||
T7277 | SB 242084 | SB 242084 dihydrochloride hydrate | 5-HT Receptor |
SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor. | |||
T8441 | Lerisetron | 5-HT Receptor | |
Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity. | |||
T1042 | Granisetron hydrochloride | BRL 43694A,Granisetron HCl | 5-HT Receptor |
Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy patients. | |||
T50011 | (2-methylpropyl)({[3-(trifluoromethyl)phenyl]methyl})amine | Others | |
(2-methylpropyl)({[3-(trifluoromethyl)phenyl]methyl})amine is a selective serotonin receptor agonist that specifically targets 5-HT2A and 5-HT2C receptors. It has been used to study the role of serotonin in a variety of ... | |||
T1173 | Tropisetron hydrochloride | SDZ-ICS 930,Tropisetron HCl,ICS 205-930 | 5-HT Receptor |
Tropisetron hydrochloride (Tropisetron HCl) is the hydrochloride salt form of tropisetron, a selective, competitive serotonin 5-hydroxytryptamine type 3 (5-HT3) receptor antagonist, with antinauseant and antiemetic activ... | |||
T1478 | Ondansetron hydrochloride dihydrate | SN 307,NSC 665799,GR 38032,Ondansetron hydrochloride | 5-HT Receptor |
Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist. It is effective in the treatment of nausea and vomiting caused by cytotoxic chemotherapy drugs, including cisplatin, a... | |||
T50089 | 2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine | Others | |
2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine is an indoleamine compound that is structurally similar to serotonin. It is a selective agonist at the 5-HT2A receptor and has potential applications in neuroscience. | |||
T50039 | 3-(2-aminopropyl)phenol hydrochloride | Others | |
3-(2-aminopropyl)phenol hydrochloride is a phenethylamine analog used as a molecular structural unit. It is a psychoactive drug that is a partial agonist at several serotonin receptors, including 5-HT1A, 5-HT1B, and 5-HT... | |||
T4429 | Rauwolscine hydrochloride | Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride | Adrenergic Receptor |
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b... | |||
T60330 | Metapramine | ||
Metapramine (19560 RP) is a tricyclic antidepressant[1]. Metapramine inhibits norepinephrine reuptake without affecting the reuptake of serotonin or dopamine [1] [2] [3]. Metapramine is a low-affinity antagonist of the N... | |||
T6S1684 | 8-Gingerol | Antioxidant , Antibacterial , TRP/TRPV Channel | |
1. 8-Gingerol has antioxidant activity. 2. 8-Gingerol has antimycobacterial activity. 3. 8-Gingerol could be used as an effective skin-whitening agent. 4. 8-Gingerol shows antipyretic and anti-inflammation characteristic... | |||
T27675 | JNJ-28583867 | JNJ28583867 | |
JNJ-28583867 is an inhibitor of histamine H(3) receptor antagonist and serotonin reuptake. | |||
T71046 | FK-1052 | ||
FK-1052 is a serotonin 3 & 4 dual receptor antagonist. | |||
T71045 | FK-1052 HCl | ||
FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist. | |||
T22340 | Granisetron | Sustol,Granisetronum,Sancuso,Kevatril | 5-HT Receptor |
Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy. | |||
T27607 | Indisetron Dihydrochloride | N3389T,Sinseron,N-3389T,N 3389T | |
Indisetron Dihydrochloride is a 5-HT(3) and 5-HT(4) receptor antagonist. Indisetron reduces 2-methyl-5-serotonin (HT)-induced bradycardia. |